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SAG Hedgehog pathway activator; Activates Smoothened (SMO)
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(S)-MG132 Ubiquitin-proteasome inhibitor; NF-kB pathway inhibitor; IκB activator
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Ruxolitinib JAK/STAT pathway inhibitor; Inhibits JAK1 and JAK2
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Rucaparib Poly ADP ribose polymerase (PARP) inhibitor
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RSC-133 Epigenetic modifier; Inhibits DNA methyltransferase (DNMT)
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Rosiglitazone PPARγ activator
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Rolipram cAMP pathway activator; Inhibits type 4 cyclic nucleotide phosphodiesterases (PDE4)
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RG108 Epigenetic modifier; Inhibits DNA methyltransferase (DNMT)
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Reversine Adenosine receptor, non-muscle myosin II (NM II), MEK1, and aurora kinase inhibitor
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Resveratrol Antioxidant; COX-1 inhibitor
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RepSox (Hydrochloride) Activin/BMP/TGF-β pathway inhibitor; Inhibits ALK5
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Refametinib MEK/ERK pathway inhibitor; Inhibits MEK1 and MEK2